SCHEMBL20060200

SCHEMBL20060200

CN(C)/C=C1/CCC(=N)/C(=C\NCc2ccccc2)C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ADH1B P00325 1/20 0.36
ADH1C P00326 1/20 0.36
ADH1A P07327 1/20 0.36
ADH7 P40394 1/20 0.36
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 3/20 0.34
HTT P42858 1/20 0.34
HIF1A Q16665 1/20 0.34
USP2 O75604 1/20 0.34
MAP1LC3B Q9GZQ8 1/20 0.32
HSD17B10 Q99714 1/20 0.30
NSD2 O96028 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20060210 0.80
SCHEMBL20060197 0.78
SCHEMBL20060185 0.77
SCHEMBL20060150 0.76 KDM4E (0.31) KMT2AKDM4EMEN1
SCHEMBL20060207 0.72 KMT2A (0.35) KMT2AALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL20060208 0.71 KDM4E (0.34) KMT2AALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL20060035 0.67 KDM4E (0.36) KMT2AALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL20060212 0.66 MAPT (0.32) KMT2AALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL11665421 0.65 ADH1B (0.50) KMT2AALDH1A1SMN1; SMN2L3MBTL1ADH1B
SCHEMBL1309772 0.63 KMT2A (0.94) KMT2AALDH1A1SMN1; SMN2L3MBTL1ADH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed