SCHEMBL2006062

SCHEMBL2006062

O=C(c1nc(-c2cccnc2)no1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
GAA P10253 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
GSK3B P49841 4/20 0.43
PTGES2 Q9H7Z7 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HDAC6 Q9UBN7 3/20 0.37
HDAC1 Q13547 2/20 0.37
TBXAS1 P24557 1/20 0.37
MAPT P10636 2/20 0.37
F2 P00734 1/20 0.37
F12 P00748 1/20 0.37
KLK7 P49862 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008785 0.94 GAA (0.46) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2004796 0.93 CYP1A2 (0.45) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2002528 0.92 CYP1A2 (0.48) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL1997418 0.92 CYP3A4 (0.43) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2002145 0.91 LMNA (0.43) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2004059 0.90 S1PR1 (0.46) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2000479 0.89 CYP1A2 (0.44) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2004345 0.89 SMPD1 (0.41) CYP3A4GSK3BL3MBTL1LMNATSHR
SCHEMBL2005780 0.86 LMNA (0.41) CYP1A2CYP3A4GAACYP2D6CYP2C9
SCHEMBL2003553 0.85 GSK3B (0.42) CYP1A2CYP3A4GAACYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed