SCHEMBL2006192

SCHEMBL2006192

Cc1c(CC(=O)O)c2c(F)c(O)ccc2n1C(=O)C1CCN(C)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.35
AKR1C3 P42330 4/20 0.34
AKR1C2 P52895 4/20 0.34
ALDH1A1 P00352 3/20 0.34
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
KDM4A O75164 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
TSHR P16473 2/20 0.32
POLB P06746 1/20 0.32
GRM5 P41594 1/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.31
PTGIR P43119 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
NFKB1 P19838 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005629 0.90 AKR1C3 (0.36) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL2008383 0.90 AKR1C3 (0.36) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL2009474 0.89 PTGDR2 (0.37) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL2008214 0.88 AKR1C3 (0.35) RIPK1AKR1C3AKR1C2PTGS1PTGS2
SCHEMBL2003676 0.88 PTGS1 (0.38) RIPK1AKR1C3AKR1C2ALDH1A1GAA
SCHEMBL2004832 0.87 AKR1C3 (0.36) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL2005105 0.87 AKR1C3 (0.34) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL2002989 0.87 PTGDR2 (0.39) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL2002210 0.83 GAA (0.36) AKR1C3AKR1C2ALDH1A1GAAMAPT
SCHEMBL2008035 0.81 AKR1C3 (0.39) AKR1C3AKR1C2ALDH1A1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed