SCHEMBL2002210

SCHEMBL2002210

Cc1c(CC(=O)O)c2c(F)c(O)ccc2n1C(=O)N1CCN(C)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
AKR1C3 P42330 6/20 0.35
AKR1C2 P52895 6/20 0.35
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34
CNR2 P34972 1/20 0.33
PTGDR2 Q9Y5Y4 3/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
HIF1A Q16665 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PTGDR Q13258 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006737 0.90 CNR2 (0.38) GAAALDH1A1AKR1C3AKR1C2PTGS1
SCHEMBL2005004 0.88 REN (0.37) AKR1C3AKR1C2PTGS1PTGS2CNR2
SCHEMBL2000853 0.87 GAA (0.39) GAAALDH1A1MAPTAKR1C3AKR1C2
SCHEMBL2005243 0.86 AKR1C3 (0.39) GAAALDH1A1MAPTAKR1C3AKR1C2
SCHEMBL2006192 0.83 RIPK1 (0.35) GAAALDH1A1MAPTAKR1C3AKR1C2
SCHEMBL2005126 0.80 AKR1C3 (0.40) AKR1C3AKR1C2PTGS1PTGS2CNR2
SCHEMBL12255389 0.78 GAA (0.41) GAAALDH1A1MAPTAKR1C3AKR1C2
SCHEMBL2005937 0.78 PTGS1 (0.40) ALDH1A1MAPTAKR1C3AKR1C2PTGS1
SCHEMBL2003517 0.77 PTGS1 (0.57) MAPTAKR1C3AKR1C2PTGS1PTGS2
SCHEMBL2005629 0.76 AKR1C3 (0.36) AKR1C3AKR1C2PTGS1PTGS2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed