SCHEMBL20063802

SCHEMBL20063802

Bc1nc(N)c2nc(C)n(CC)c2n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.38
ADORA2A P29274 4/20 0.38
ADORA1 P30542 4/20 0.38
ADORA2B P29275 3/20 0.38
KDM4E B2RXH2 1/20 0.34
RAD52 P43351 1/20 0.34
TLR7 Q9NYK1 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
ALDH1A1 P00352 2/20 0.31
GAA P10253 2/20 0.31
MAPT P10636 2/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21242920 0.84 ADORA2A (0.39) ADORA3ADORA2AADORA1ADORA2BCDK1
SCHEMBL13727333 0.82 ADORA2A (0.41) ADORA3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL13233221 0.77 ADORA2A (0.49) ADORA3ADORA2AADORA1ADORA2BTLR7
SCHEMBL13091617 0.71 CDK1 (0.38) ADORA3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL21242911 0.67 ADORA2A (0.37) ADORA3ADORA2AADORA1ADORA2BCDK1
SCHEMBL10309720 0.66 ADORA1 (0.40) ADORA3ADORA2AADORA1ADORA2BTLR7
SCHEMBL10121588 0.63 ADORA2A (0.38) ADORA3ADORA2AADORA1ADORA2BTLR7
SCHEMBL5391550 0.63 CDK1 (0.47) ADORA3ADORA2AADORA1ADORA2BTLR7
SCHEMBL12028042 0.61 ADORA2A (0.59) ADORA3ADORA2AADORA1ADORA2BCDK1
SCHEMBL20759785 0.61 ADORA3 (0.37) ADORA3ADORA2AADORA1ADORA2BCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071531-A1 HPPK INHIBITORS USEFUL AS ANTIBACTERIAL AGENTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2018-04-19 WO disclosed