SCHEMBL20064053

SCHEMBL20064053

O=CNC1CN(c2ccccn2)C1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.46
GRIN2B Q13224 4/20 0.44
GRM1 Q13255 5/20 0.44
PLD1 Q13393 1/20 0.44
KAT2B Q92831 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
GRM5 P41594 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 1/20 0.41
CHRM4 P08173 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13449831 0.88 CA12 (0.50) USP30GRM1PLD1KAT2BALDH1A1
SCHEMBL20065110 0.88 CA12 (0.50) USP30GRM1PLD1KAT2BALDH1A1
SCHEMBL29969592 0.78 KDM4E (0.49) USP30GRIN2BGRM1PLD1KAT2B
SCHEMBL20064228 0.77 KDM4E (0.43) GRM1KDM4ECHRM4
SCHEMBL2005995 0.76 USP30 (0.54) USP30GRIN2BGRM1CYP3A4CYP2D6
SCHEMBL20064573 0.75 GRIN2D (0.41) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7711658 0.74 HRH3 (0.48) CYP3A4ALDH1A1KDM4E
SCHEMBL20063997 0.74 USP30 (0.47) USP30CHRM4
SCHEMBL28768958 0.73 HSD11B1 (0.49) GRIN2BGRM1PLD1CYP3A4CYP2D6
SCHEMBL23875353 0.72 PLD1 (0.52) GRIN2BGRM1PLD1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed