SCHEMBL20064173

SCHEMBL20064173

CCc1cc(F)cc(OC2CCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
ALDH1A1 P00352 2/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
TSHR P16473 1/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
GRM5 P41594 2/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
ALOX12 P18054 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13534139 0.84 GRIN2D (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9913868 0.82 FFAR4 (0.44) FFAR4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL22150460 0.78 SLC6A2 (0.35) GRIN1GRIN2BCYP4F2CYP4A11SLC6A2
SCHEMBL20325313 0.78 SLC6A2 (0.33) GRIN1GRIN2BALDH1A1CYP4F2CYP4A11
SCHEMBL28014799 0.78 EPHX2 (0.42) FFAR4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL24196240 0.75 GRIN2D (0.49) FFAR4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL20064585 0.75 ALDH1A1 (0.48) ALDH1A1SLC6A2SLC6A4SLC6A3OPRK1
SCHEMBL22560560 0.74 EPHX2 (0.33) SLC6A2SLC6A4SLC6A3EPHX2OPRM1
SCHEMBL19510585 0.74 FFAR4 (0.40) FFAR4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3037790 0.73 EPHX2 (0.48) FFAR4GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed