SCHEMBL20064289

SCHEMBL20064289

CCCCCc1ccc(C)c2cccnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.50
PSMD14 O00487 2/20 0.50
COPS5 Q92905 2/20 0.50
SLC6A2 P23975 1/20 0.50
CCR1 P32246 3/20 0.42
CCR8 P51685 3/20 0.42
L3MBTL1 Q9Y468 7/20 0.42
NPC1 O15118 3/20 0.42
HSP90AA1 P07900 1/20 0.42
CCR5 P51681 2/20 0.41
KDM4E B2RXH2 5/20 0.40
BRD4 O60885 1/20 0.40
MITF O75030 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
SLC40A1 Q9NP59 1/20 0.39
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10157939 0.82 HTT (0.58) HTTPSMD14COPS5SLC6A2CCR1
SCHEMBL28423616 0.78 L3MBTL1 (0.53) HTTPSMD14COPS5SLC6A2CCR1
SCHEMBL29459602 0.78 L3MBTL1 (0.53) HTTPSMD14COPS5SLC6A2CCR1
SCHEMBL11515706 0.77 KDM4E (0.64) HTTSLC6A2L3MBTL1NPC1KDM4E
SCHEMBL31026573 0.77 L3MBTL1 (0.52) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL1416783 0.77 L3MBTL1 (0.52) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL28067774 0.77 HTT (0.56) HTTPSMD14COPS5SLC6A2CCR1
SCHEMBL31026570 0.77 L3MBTL1 (0.52) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL31026586 0.77 L3MBTL1 (0.52) CCR1CCR8L3MBTL1NPC1HSP90AA1
SCHEMBL27455037 0.76 CYP1A2 (0.50) HTTKDM4ETDP1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed