SCHEMBL20064321

SCHEMBL20064321

COc1cccc(C)c1NC(C)=S

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.49
GAA P10253 2/20 0.44
TAAR1 Q96RJ0 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
PKM P14618 1/20 0.43
LMNA P02545 1/20 0.42
S1PR2 O95136 1/20 0.41
S1PR4 O95977 1/20 0.41
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
S1PR5 Q9H228 1/20 0.41
ALDH1A1 P00352 3/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
KMT2A Q03164 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19573888 0.89 KMT2A (0.45) ATMGAACYP3A4LMNAALDH1A1
SCHEMBL16119698 0.84 ATM (0.48) ATMGAATAAR1CYP1A2CYP3A4
SCHEMBL12627891 0.82 LMNA (0.52) ATMGAACYP1A2CYP2C19LMNA
SCHEMBL5480782 0.82 ATM (0.56) ATMCYP1A2CYP3A4CYP2C19PKM
SCHEMBL21222487 0.81 HPGD (0.51) GAALMNAALDH1A1KMT2AL3MBTL1
SCHEMBL24834185 0.77 ATM (0.48) ATMGAATAAR1CYP1A2CYP3A4
SCHEMBL11142783 0.77 ATM (0.45) ATMGAACYP1A2CYP3A4CYP2C19
SCHEMBL11664862 0.75 TAAR1 (0.49) ATMTAAR1CYP1A2CYP3A4CYP2C19
SCHEMBL15484253 0.75 HPGD (0.51) GAACYP3A4LMNAALDH1A1KMT2A
SCHEMBL15883199 0.75 ALDH1A1 (0.55) ATMTAAR1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed