SCHEMBL20064340

SCHEMBL20064340

CNc1c(C)cccc1OC1CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
EPHX2 P34913 2/20 0.39
HRH1 P35367 2/20 0.38
CARM1 Q86X55 1/20 0.37
PRMT1 Q99873 1/20 0.37
MCHR1 Q99705 3/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 1/20 0.37
HTR1A P08908 1/20 0.37
KAT2B Q92831 1/20 0.36
BAZ2B Q9UIF8 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR1B P28222 1/20 0.36
CXCR5 P32302 1/20 0.36
ALOX12 P18054 1/20 0.36
EPHX1 P07099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31448456 0.80 MCHR1 (0.40) PDE4APDE4BPDE4CPDE4DCARM1
SCHEMBL31448546 0.79 MCHR1 (0.42) PDE4APDE4BPDE4CPDE4DCARM1
SCHEMBL28331538 0.79 PDE4D (0.50) PDE4APDE4BPDE4CPDE4DCARM1
SCHEMBL13696497 0.78 SLC6A2 (0.49) EPHX2HRH1SLC6A2SLC6A4SLC6A3
SCHEMBL7701922 0.74 SLC6A2 (0.49) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL29952646 0.74 TLR2 (0.39) EPHX2HRH1MCHR1KAT2BBAZ2B
SCHEMBL15057752 0.74 MRGPRX1 (0.43) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL11586746 0.74 MCHR1 (0.46) PDE4APDE4BPDE4CPDE4DCARM1
SCHEMBL10525480 0.73 SLC6A2 (0.47) EPHX2CARM1PRMT1MCHR1SLC6A2
SCHEMBL1006539 0.73 CYP1A2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed