SCHEMBL20064397

SCHEMBL20064397

Cc1cnc(N2CC(NC=O)C2)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.39
GPR119 Q8TDV5 2/20 0.36
ADH1B P00325 3/20 0.33
ADH1A P07327 3/20 0.33
OPRK1 P41145 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
MAPK1 P28482 1/20 0.33
CHRM4 P08173 2/20 0.32
ACKR3 P25106 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20064573 0.80 GRIN2D (0.41) GPR119HDAC6SLC6A9
SCHEMBL20064017 0.79 HRH4 (0.44) ACACBGPR119MAPK1KCNH2
SCHEMBL17972943 0.72 TSHR (0.39) ACACBGPR119HDAC6MAPK1KCNH2
SCHEMBL16472351 0.72 ACACB (0.39) ACACBGPR119OPRK1HDAC6MAPK1
SCHEMBL17973025 0.71 HRH3 (0.41) ACACBGPR119KCNH2SLC6A9AOC3
SCHEMBL12457553 0.71 ACACB (0.41) ACACBGPR119HDAC6KCNH2SLC6A9
SCHEMBL24962247 0.70 ACACB (0.39) ACACBGPR119MAPK1KCNH2SLC6A9
SCHEMBL21227806 0.69 JAK3 (0.45) ACACB
SCHEMBL16302107 0.69 KDM4E (0.45) ACACBGPR119HDAC3HDAC4HDAC1
SCHEMBL12490730 0.69 OPRK1 (0.52) GPR119OPRK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed