SCHEMBL20064017

SCHEMBL20064017

CNC1CN(c2ncc(C)cn2)C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 12/20 0.44
HRH3 Q9Y5N1 9/20 0.41
ACACB O00763 1/20 0.39
GPR119 Q8TDV5 1/20 0.36
HRH1 P35367 3/20 0.36
KCNH2 Q12809 2/20 0.36
HRH2 P25021 2/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20283137 0.83 CHRM4 (0.41) HRH4HRH3HRH1KCNH2HRH2
SCHEMBL12525108 0.81 GPR119 (0.47) HRH4GPR119KCNH2MAPK1
SCHEMBL20064080 0.80 HRH3 (0.40) HRH4HRH3
SCHEMBL24964199 0.79 HRH4 (0.53) HRH4HRH3
SCHEMBL20283121 0.79 CHRM4 (0.47) HRH4ACACB
SCHEMBL20064397 0.79 ACACB (0.39) ACACBGPR119KCNH2MAPK1
SCHEMBL17972943 0.78 TSHR (0.39) ACACBGPR119KCNH2MAPK1
SCHEMBL16472351 0.78 ACACB (0.39) ACACBGPR119KCNH2MAPK1
SCHEMBL19604915 0.77 HRH3 (0.45) HRH4HRH3GPR119KCNH2
SCHEMBL20283122 0.76 ACACB (0.49) HRH4HRH3ACACBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed