Pefurazoate

Pefurazoate

SCHEMBL20067

C=CCCCOC(=O)C(CC)N(Cc1ccco1)C(=O)n1ccnc1

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.35
TSHR P16473 4/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP2C9 P11712 1/20 0.34
NPSR1 Q6W5P4 4/20 0.33
ALDH1A1 P00352 5/20 0.33
MAPK1 P28482 2/20 0.33
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
TBXA2R P21731 1/20 0.33
POLB P06746 1/20 0.33
USP2 O75604 1/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
GAA P10253 1/20 0.31
TP53 P04637 1/20 0.31
FNTA P49354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R)-(+)-Pefurazoate SCHEMBL8163178 1.00 MAPT (0.35) MAPTTSHRCYP1A2CYP3A4CYP2C19
Pefurazoate SCHEMBL27797684 0.99 MAPT (0.35) MAPTTSHRCYP1A2CYP3A4CYP2C19
Pefurazoate SCHEMBL28180407 0.93 MAPT (0.32) MAPTTSHRCYP1A2CYP3A4CYP2C19
Pefurazoate SCHEMBL28269053 0.91 POLB (0.33) MAPTTSHRCYP1A2CYP3A4CYP2C19
SCHEMBL28641743 0.85 TSHR (0.36) MAPTTSHRCYP1A2CYP3A4CYP2C19
SCHEMBL19186469 0.85 MAPT (0.34) MAPTTSHRCYP1A2CYP3A4CYP2C19
Pefurazoate SCHEMBL4284449 0.84 IDO1 (0.51) MAPTTSHRCYP1A2CYP3A4CYP2C19
Pefurazoate SCHEMBL6433092 0.83 TSHR (0.35) MAPTTSHRCYP1A2CYP3A4CYP2C19
Pefurazoate SCHEMBL28785223 0.83 MEN1 (0.45) MAPTPOLBTDP1TP53
SCHEMBL21093425 0.82 TBXA2R (0.39) TSHRCYP1A2CYP3A4CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 20712 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
US-20260137082-A1 FUNGICIDAL COMPOSITIONS COMPRISING FLUDIOXONIL SYNGENTA CROP PROTECTION AG (CH) 2026-05-21 US claimed
CN-120008044-B System and method for evaluating state of incinerator for salt-containing chlorine-containing waste liquid 江苏瑞鼎环境工程有限公司 2026-05-12 CN claimed
US-20260101893-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-04-16 US claimed
US-20260076366-A1 SYNERGISTIC PESTICIDAL COMPOSITIONS AND METHODS FOR DELIVERY OF ACTIVE INGREDIENTS 0903608 B C LTD (CA) 2026-03-19 US claimed
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
US-20260068884-A1 COMPOSITION USED FOR KILLING FUNGI AND METHOD FOR APPLYING COMPOSITION JIANGSU FLAG CHEMICAL INDUSTRY CO., LTD. (CN) 2026-03-12 US claimed
WO-2026041871-A1 METHODS OF CONTROLLING CAUSAL AGENTS OF RAMULARIA LEAF SPOT OR RHYNCHOSPORIUM LEAF SCALD DISEASE, AND COMPOSITIONS FOR THE SAME GOWAN CROP PROTECTION LIMITED (GB) 2026-02-26 WO claimed
EP-4114183-B1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-02-25 EP claimed
US-RE50724-E1 4-membered ring carboxamides used as nematicides SYNGENTA CROP PROTECTION AG (CH) 2026-01-06 US claimed
EP-0827553-A1 COMBINATIONS OF ACTIVE SUBSTANCES BAYER AG (DE) 1998-03-11 EP claimed
EP-0609099-B1 Antimicrobial and antifungal compositions comprising silicon-compounds, and their use in agriculture and horticulture SANKYO CO (JP) 1997-03-26 EP claimed
WO-1996036739-A1 COMBINATIONS OF ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 1996-11-21 WO claimed
EP-0734650-A2 Patch preparations for treating plants NIHON BAYER AGROCHEM K.K. (JP) 1996-10-02 EP claimed
US-5500437-A SYNERGISTIC COMBINATION TO PROTECT CEREAL PLANTS AND SEEDS FROM PLANT DISEASES CIBA-GEIGY, AG (CH) 1996-03-19 US claimed
US-5468747-A Fungicidal compositions and methods of use employing pyrimidine derivatives ZENECA LIMITED (GB) 1995-11-21 US claimed
EP-0603845-B1 Fungicide composition for agriculture and horticulture KUREHA CHEMICAL IND CO LTD (JP) 1995-11-02 EP claimed
EP-0613619-A1 Microbicides CIBA-GEIGY AG (CH) 1994-09-07 EP claimed
EP-0609099-A1 Antimicrobial and antifungal compositions comprising silicon-compounds, and their use in agriculture and horticulture SANKYO COMPANY LIMITED (JP) 1994-08-03 EP claimed
EP-0603845-A1 Fungicide composition for agriculture and horticulture KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1994-06-29 EP claimed