SCHEMBL20074069

SCHEMBL20074069

CC[C@@]1(C(=O)N(C)CCCC2CCN(c3ccc(C(=O)N(C)C)c(Cl)n3)CC2)CCOC1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 7/20 0.32
GPR119 Q8TDV5 4/20 0.32
ACACB O00763 2/20 0.32
ACACA Q13085 2/20 0.32
NAPEPLD Q6IQ20 4/20 0.32
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20072053 0.87 ACACB (0.36) ACACBACACANAPEPLDALDH1A1
SCHEMBL20072052 0.87 ACACB (0.36) ACACBACACANAPEPLDALDH1A1
SCHEMBL21644274 0.87 ACACB (0.36) ACACBACACANAPEPLDALDH1A1
SCHEMBL20072200 0.84 TSHR (0.37) ACACBACACANAPEPLDALDH1A1
SCHEMBL20072009 0.83 GPR119 (0.38) TPH1GPR119ACACBACACAMEN1
SCHEMBL21644270 0.81 GPR119 (0.37) GPR119
SCHEMBL20072011 0.81 GPR119 (0.37) GPR119ACACBACACAMEN1KMT2A
SCHEMBL21644279 0.81 GPR119 (0.37) GPR119ACACBACACAMEN1KMT2A
SCHEMBL20072202 0.81 GPR119 (0.37) GPR119
SCHEMBL20072010 0.81 GPR119 (0.37) GPR119ACACBACACAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071313-A1 N-ARYL AND N-HETEROARYL PIPERIDINE DERIVATIVES AS LIVER X RECEPTOR BETA AGONISTS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME CORP. (US) 2018-04-19 WO disclosed