Asalhydromorphone

Asalhydromorphone

SCHEMBL20077472

CC(=O)Oc1ccccc1C(=O)OC1=CCC2C3Cc4ccc(OC(=O)c5ccccc5OC(C)=O)c5c4C2(CCN3C)C1O5

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 11/20 0.53
OPRM1 P35372 7/20 0.49
OPRK1 P41145 5/20 0.49
MRGPRX2 Q96LB1 2/20 0.49
LMNA P02545 1/20 0.49
PDE4D Q08499 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Asalhydromorphone SCHEMBL31237072 1.00 OPRD1 (0.53) OPRD1OPRM1OPRK1MRGPRX2LMNA
Asalhydromorphone SCHEMBL15028750 1.00 OPRD1 (0.53) OPRD1OPRM1OPRK1MRGPRX2LMNA
SCHEMBL20077628 0.95 OPRD1 (0.48) OPRD1OPRM1OPRK1MRGPRX2LMNA
SCHEMBL20077473 0.93 OPRD1 (0.49) OPRD1OPRM1OPRK1MRGPRX2LMNA
SCHEMBL16922127 0.91 OPRD1 (0.59) OPRD1OPRM1OPRK1MRGPRX2LMNA
SCHEMBL20077664 0.88 OPRD1 (0.51) OPRD1OPRM1OPRK1MRGPRX2LMNA
SCHEMBL15028743 0.87 OPRD1 (0.49) OPRD1OPRM1OPRK1MRGPRX2LMNA
SCHEMBL20077663 0.86 OPRD1 (0.52) OPRD1OPRM1OPRK1MRGPRX2LMNA
Thebacon SCHEMBL21304123 0.86 OPRD1 (0.63) OPRD1OPRM1OPRK1MRGPRX2LMNA
Thebacon SCHEMBL1649199 0.86 OPRD1 (0.63) OPRD1OPRM1OPRK1MRGPRX2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200038383-A1 IMMEDIATE-RELEASE ABUSE DETERRENT COMPOSITIONS OR MEDICAMENTS FOR TREATING PAIN, ADD, ADHD AND OTHER SYNDROMES OR DISORDERS ALTER DOMUS (US) LLC 2020-02-06 US disclosed
WO-2018071879-A1 IMMEDIATE-RELEASE ABUSE DETERRENT COMPOSITIONS OR MEDICAMENTS FOR TREATING PAIN, ADD, ADHD AND OTHER SYNDROMES OR DISORDERS KEMPHARM, INC. (US) 2018-04-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200038383-A1 IMMEDIATE-RELEASE ABUSE DETERRENT COMPOSITIONS OR MEDICAMENTS FOR TREATING PAIN, ADD, ADHD AND OTHER SYNDROMES OR DISORDERS OPRK1, OPRL1, OPRD1 OPRD1 3/4885OPRM1 4/4885OPRK1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.