SCHEMBL20079900

SCHEMBL20079900

c1ccc2c(c1)OC(c1ccc3c(c1)OCC3)O2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ITGB2 P05107 1/20 0.38
ICAM1 P05362 1/20 0.38
ITGAL P20701 1/20 0.38
NOTUM Q6P988 1/20 0.38
KDM1A O60341 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
LMNA P02545 2/20 0.34
CRHBP P24387 2/20 0.34
CRHR2 Q13324 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HTT P42858 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRM3 P20309 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18896908 0.78 NPC1 (0.32) NPC1RAB9ASMN1; SMN2ESR1ESR2
SCHEMBL24317332 0.76 ALOX15 (0.51) NPC1RAB9AITGB2ICAM1ITGAL
SCHEMBL20846975 0.74 KDM4E (0.48) CYP1A2NPC1RAB9AKDM1AMAOA
SCHEMBL22221860 0.73 RAB9A (0.53) NPC1RAB9AITGB2ICAM1ITGAL
SCHEMBL335161 0.71
SCHEMBL33192 0.71
SCHEMBL29373453 0.71
SCHEMBL11480538 0.71 EPHX2 (0.40) CYP1A2SMN1; SMN2
SCHEMBL19346223 0.70 ALOX15 (0.51) NPC1RAB9AITGB2ICAM1ITGAL
SCHEMBL25901189 0.70 RAB9A (0.50) NPC1RAB9AMAOBESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3915367-A1 DIKETONES AND HYDROXYKETONES AS CATENIN SIGNALING PATHWAY ACTIVATORS BioSplice Therapeutics, Inc. (US) 2021-12-01 EP disclosed
EP-3311666-B1 DIKETONES AND HYDROXYKETONES AS CATENIN SIGNALING PATHWAY ACTIVATORS SAMUMED LLC (US) 2021-05-05 EP disclosed
EP-3311666-A1 DIKETONES AND HYDROXYKETONES AS CATENIN SIGNALING PATHWAY ACTIVATORS Samumed, LLC (US) 2018-04-25 EP disclosed