SCHEMBL2008138

SCHEMBL2008138

COc1ccc2c(c1)c(CC(=O)O)c(C)n2C(=O)c1ccccn1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.73
CYP1A2 P05177 2/20 0.73
CYP2D6 P10635 2/20 0.73
CYP2C9 P11712 2/20 0.73
HIF1A Q16665 2/20 0.73
NPSR1 Q6W5P4 2/20 0.73
TSHR P16473 1/20 0.73
NFKB1 P19838 1/20 0.73
AKR1C3 P42330 8/20 0.68
AKR1C2 P52895 7/20 0.68
AKR1C4 P17516 2/20 0.63
AKR1C1 Q04828 2/20 0.63
PTGS2 P35354 2/20 0.63
KDM4E B2RXH2 1/20 0.63
MEN1 O00255 1/20 0.63
PTGES O14684 1/20 0.63
ABCC3 O15438 1/20 0.63
ABCC4 O15439 1/20 0.63
ABCB11 O95342 1/20 0.63
MT-CO2 P00403 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008114 0.86 PTGS1 (0.61) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL1082631 0.85 HIF1A (1.00) LMNACYP1A2CYP2D6CYP2C9HIF1A
Hydrochloric Acid SCHEMBL8646699 0.84 HIF1A (0.98) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL2005980 0.83 PTGS1 (0.67) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL2004590 0.83 PTGS1 (0.52) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL11849615 0.82 AKR1C3 (0.67) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL2008480 0.82 AKR1C3 (0.83) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL11858954 0.82 AKR1C3 (0.70) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL8645594 0.81 AKR1C3 (1.00) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL5646377 0.81 HIF1A (0.87) LMNACYP1A2CYP2D6CYP2C9HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed