SCHEMBL2008480

SCHEMBL2008480

COc1ccc2c(c1)c(CC(=O)O)c(C)n2C(=O)c1ccncc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.83
AKR1C2 P52895 8/20 0.83
HIF1A Q16665 3/20 0.81
LMNA P02545 2/20 0.81
CYP1A2 P05177 2/20 0.81
CYP2D6 P10635 2/20 0.81
CYP2C9 P11712 2/20 0.81
NPSR1 Q6W5P4 2/20 0.81
TSHR P16473 1/20 0.81
NFKB1 P19838 1/20 0.81
AKR1C4 P17516 2/20 0.77
AKR1C1 Q04828 2/20 0.77
ABCB1 P08183 2/20 0.77
PTGS1 P23219 2/20 0.77
PTGS2 P35354 2/20 0.77
GLO1 Q04760 2/20 0.77
KDM4E B2RXH2 1/20 0.77
MEN1 O00255 1/20 0.77
PTGES O14684 1/20 0.77
ABCC3 O15438 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8645594 0.91 AKR1C3 (1.00) AKR1C3AKR1C2HIF1ALMNACYP1A2
SCHEMBL1082631 0.90 HIF1A (1.00) AKR1C3AKR1C2HIF1ALMNACYP1A2
Hydrochloric Acid SCHEMBL8646699 0.89 HIF1A (0.98) AKR1C3AKR1C2HIF1ALMNACYP1A2
SCHEMBL2600801 0.89 AKR1C3 (1.00) AKR1C3AKR1C2HIF1ALMNACYP1A2
SCHEMBL12747878 0.88 AKR1C3 (0.89) AKR1C3AKR1C2HIF1ALMNACYP1A2
Niometacin SCHEMBL2010371 0.87 LMNA (0.78) AKR1C3AKR1C2HIF1ALMNACYP1A2
SCHEMBL5379167 0.87 AKR1C3 (0.83) AKR1C3AKR1C2HIF1ALMNACYP1A2
Iodoindomethacin SCHEMBL13290295 0.87 AKR1C3 (0.87) AKR1C3AKR1C2HIF1ALMNACYP1A2
Indomethacin SCHEMBL9300 0.87 PTGS2 (1.00) AKR1C3AKR1C2HIF1ALMNACYP1A2
SCHEMBL5796934 0.87 AKR1C3 (1.00) AKR1C3AKR1C2HIF1ALMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed