SCHEMBL20095307

SCHEMBL20095307

CNc1cccc(C(=O)N(C)CCON(C(=O)CCCCCCNC(=O)Nc2ccncc2)C2CCCCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 11/20 0.43
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
KEAP1 Q14145 2/20 0.36
NFE2L2 Q16236 2/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
CDK4 P11802 1/20 0.35
CCND3 P30281 1/20 0.35
PRMT3 O60678 1/20 0.35
PDE4A P27815 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27008596 0.93 NAMPT (0.43) NAMPTALDH1A1LMNAKEAP1NFE2L2
SCHEMBL20095389 0.91 NAMPT (0.43) NAMPTALDH1A1LMNAKEAP1NFE2L2
SCHEMBL30292608 0.90 NAMPT (0.41) NAMPTALDH1A1LMNAKEAP1NFE2L2
SCHEMBL20095455 0.90 NAMPT (0.41) NAMPTALDH1A1LMNAKEAP1NFE2L2
SCHEMBL20095473 0.83 NAMPT (0.51) NAMPTALDH1A1LMNAKEAP1NFE2L2
SCHEMBL20095436 0.82 NAMPT (0.46) NAMPTALDH1A1LMNAKEAP1NFE2L2
SCHEMBL20095426 0.80 NAMPT (0.47) NAMPTPDE4A
SCHEMBL20095298 0.80 NAMPT (0.47) NAMPTPDE4A
SCHEMBL21471208 0.76 NAMPT (0.32) NAMPTPDE4A
SCHEMBL20095369 0.76 NAMPT (0.32) NAMPTPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240016953-A1 TARGETED DELIVERY OF NICOTINAMINDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITORS SEAGEN INC (US) 2024-01-18 US disclosed
US-20240016953-A1 TARGETED DELIVERY OF NICOTINAMINDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITORS SEAGEN INC (US) 2024-01-18 US disclosed
US-11638762-B2 Targeted delivery of nicotinamide adenine dinucleotide salvage pathway inhibitors SEAGEN INC. (US) 2023-05-02 US disclosed
US-20190314519-A1 TARGETED DELIVERY OF NICOTINAMIDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITORS SEATTLE GENETICS, INC. (US) 2019-10-17 US disclosed
WO-2018075600-A1 TARGETED DELIVERY OF NICOTINAMIDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITORS SEATTLE GENETICS, INC. (US) 2018-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240016953-A1 TARGETED DELIVERY OF NICOTINAMINDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITORS NAMPT, NAPRT, NNMT NAMPT 1/4885ALDH1A1 2101/4885LMNA 1489/4885
US-20190314519-A1 TARGETED DELIVERY OF NICOTINAMIDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITORS NAMPT, NME4, NNMT NAMPT 1/4885ALDH1A1 2315/4885LMNA 1619/4885
US-11638762-B2 Targeted delivery of nicotinamide adenine dinucleotide salvage pathway inhibitors NAMPT, NME4, NNMT NAMPT 1/4885ALDH1A1 2315/4885LMNA 1619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.