SCHEMBL2009534

SCHEMBL2009534

COc1cc2c(CC(=O)O)c(C)n(C(=O)c3cccnc3)c2cc1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.56
PTGS1 P23219 2/20 0.56
LMNA P02545 2/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2D6 P10635 2/20 0.54
CYP2C9 P11712 2/20 0.54
HIF1A Q16665 2/20 0.54
NPSR1 Q6W5P4 2/20 0.54
TSHR P16473 1/20 0.54
NFKB1 P19838 1/20 0.54
AKR1C3 P42330 9/20 0.52
AKR1C2 P52895 9/20 0.52
ABCB1 P08183 3/20 0.47
PTGDR2 Q9Y5Y4 2/20 0.47
AKR1C4 P17516 2/20 0.47
AKR1C1 Q04828 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
PTGES O14684 1/20 0.47
ABCC3 O15438 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5444320 0.89 LMNA (0.67) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL2006282 0.89 PTGS2 (0.72) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL2007832 0.88 PTGS1 (0.62) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL2002636 0.87 AKR1C3 (0.49) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL3002102 0.84 AKR1C3 (0.72) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL5433909 0.84 AKR1C3 (0.68) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL2002963 0.83 LMNA (0.48) PTGS2PTGS1LMNACYP1A2CYP2D6
Niometacin SCHEMBL2010371 0.83 LMNA (0.78) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL5452320 0.83 AKR1C3 (0.72) PTGS2PTGS1LMNACYP1A2CYP2D6
SCHEMBL5448589 0.83 PTGS1 (0.66) PTGS2PTGS1LMNACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed