SCHEMBL20095940

SCHEMBL20095940

CC(C)(C)OC(=O)NC1CC(F)(F)CC[C@@H]1NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.40
RORC P51449 2/20 0.39
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
CTSK P43235 2/20 0.38
KDM1A O60341 2/20 0.37
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MAOB P27338 2/20 0.36
MAOA P21397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20063805 1.00 BTK (0.40) BTKRORCNFKB1NFKB2RELA
SCHEMBL1992927 0.89 NFKB1 (0.42) BTKNFKB1NFKB2RELACTSK
SCHEMBL15420557 0.87 BTK (0.47) BTKRORCNFKB1NFKB2RELA
SCHEMBL15420433 0.87 BTK (0.47) BTKRORCNFKB1NFKB2RELA
SCHEMBL20959100 0.87 BTK (0.47) BTKRORCNFKB1NFKB2RELA
SCHEMBL15420199 0.87 BTK (0.47) BTKRORCNFKB1NFKB2RELA
SCHEMBL12989321 0.87 BTK (0.47) BTKRORCNFKB1NFKB2RELA
SCHEMBL30565067 0.87 BTK (0.47) BTKRORCNFKB1NFKB2RELA
SCHEMBL15420108 0.84 RORC (0.36) BTKRORCNFKB1NFKB2RELA
SCHEMBL26253780 0.84 RORC (0.36) BTKRORCNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018072602-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2018-04-26 WO disclosed