SCHEMBL20100285

SCHEMBL20100285

COC(=O)c1ccn2c1C(=O)NCC2C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.38
MAPT P10636 2/20 0.37
CDK5 Q00535 3/20 0.36
CDK5R1 Q15078 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 3/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 3/20 0.35
GAA P10253 2/20 0.35
GLA P06280 1/20 0.35
BRD4 O60885 1/20 0.35
MAPKAPK2 P49137 1/20 0.34
MAP2K1 Q02750 1/20 0.34
POLB P06746 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17485549 0.75 HTR2C (0.38) PARP1MAPTALDH1A1TSHRHPGD
SCHEMBL20100561 0.71 PARP1 (0.56) PARP1MAPTALDH1A1HSD17B10KDM4E
SCHEMBL19181725 0.64 PIK3C3 (0.37) ALDH1A1
SCHEMBL26541546 0.63 MEN1 (0.37) CDK5SMN1; SMN2KDM4EMAPKAPK2MEN1
SCHEMBL31569523 0.63 HRH3 (0.38) PARP1ALDH1A1GAA
SCHEMBL16669939 0.62 PLAT (0.39) PARP1TSHRHPGDKDM4EGAA
SCHEMBL65823 0.59 MEN1 (0.33) LMNAMEN1KMT2A
SCHEMBL16684902 0.58 ALOX5 (0.43) ALDH1A1TSHRLMNAHPGDHSD17B10
SCHEMBL17707989 0.58 PIK3C3 (0.34)
Dimethyl Phthalate SCHEMBL28064028 0.57 TSHR (0.71) MAPTALDH1A1TSHRLMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018079628-A1 PYRROLE DERIVATIVE WITH FUSED RING AND PHARMACEUTICAL USE THEREOF 大日本住友製薬株式会社 2018-05-03 WO disclosed