SCHEMBL20100593

SCHEMBL20100593

O=C(O)c1ccn2c1C(=O)NCC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
GAA P10253 2/20 0.46
PARP1 P09874 12/20 0.42
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
DAPK3 O43293 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
ABL1 P00519 1/20 0.37
NTRK1 P04629 1/20 0.37
RET P07949 1/20 0.37
MET P08581 1/20 0.37
PIM1 P11309 1/20 0.37
FGFR1 P11362 1/20 0.37
PDGFRA P16234 1/20 0.37
PRKACA P17612 1/20 0.37
FLT1 P17948 1/20 0.37
LTK P29376 1/20 0.37
GRK5 P34947 1/20 0.37
MAPK8 P45983 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20100677 0.83 ALDH1A1 (0.43) ALDH1A1GAAPARP1KDM4E
SCHEMBL20100561 0.81 PARP1 (0.56) ALDH1A1GAAPARP1KDM4EHSD17B10
SCHEMBL2485535 0.77 ALDH1A1 (0.50) ALDH1A1GAAPARP1
SCHEMBL10446487 0.75 ALDH1A1 (0.47) ALDH1A1GAAPARP1KDM4E
SCHEMBL13589774 0.74 ALDH1A1 (0.50) ALDH1A1GAAPARP1
SCHEMBL31750298 0.74 ALDH1A1 (0.50) ALDH1A1GAAPARP1KDM4E
SCHEMBL13589780 0.74 ALDH1A1 (0.50) ALDH1A1GAAPARP1
SCHEMBL20100521 0.74 ALDH1A1 (0.50) ALDH1A1GAAPARP1
SCHEMBL20123424 0.73 PARP1 (0.40) ALDH1A1GAAPARP1CHEK1AURKA
SCHEMBL20100606 0.72 RPS6KA3 (0.51) ALDH1A1GSK3BRPS6KA3KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018079628-A1 PYRROLE DERIVATIVE WITH FUSED RING AND PHARMACEUTICAL USE THEREOF 大日本住友製薬株式会社 2018-05-03 WO disclosed