SCHEMBL2010225

SCHEMBL2010225

[NH]c1ncnc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.56
PI4K2B Q8TCG2 1/20 0.56
PI4K2A Q9BTU6 1/20 0.56
PI4KB Q9UBF8 1/20 0.56
PDE4A P27815 1/20 0.56
PDE4B Q07343 1/20 0.56
PDE4C Q08493 1/20 0.56
PDE4D Q08499 1/20 0.56
ADORA2A P29274 2/20 0.52
HTT P42858 2/20 0.47
ALDH1A1 P00352 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
EGFR P00533 3/20 0.47
ABCG2 Q9UNQ0 2/20 0.47
DAPK3 O43293 1/20 0.47
MAP4K4 O95819 1/20 0.47
ABL1 P00519 1/20 0.47
ERBB2 P04626 1/20 0.47
PIM1 P11309 1/20 0.47
PRKACA P17612 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3075421 0.75 ADORA2A (0.75) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL637552 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL637551 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL3992023 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
4-Aminoquinazoline SCHEMBL142513 0.71 PI4KA (1.00) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL3951708 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL25620 0.71 PDE4A (1.00) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL11821044 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL276986 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL18087089 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103788085-A 2-(quinazoline-4-amino)-5-thiazole carboxamide derivatives and biological medicine use thereof UNIV FUDAN 2014-05-14 CN claimed
CN-103784450-A Micromolecular compound for inhibiting Src nonreceptor tyrosine kinase and pharmaceutical use thereof UNIV FUDAN 2014-05-14 CN claimed
CN-103420923-A 4-aminoquinazolinehydroxamic acid compounds and applications thereof as antitumor medicaments SINOPHARM YIXIN PHARMACEUTICAL CO LTD 2013-12-04 CN claimed
CN-101857588-A 4-aromatic aminoquinazoline derivative and purpose thereof UNIV SOUTHEAST 2010-10-13 CN claimed
EP-1976829-A2 N-(6-MEMBERED AROMATIC RING)-AMIDO ANTI-VIRAL COMPOUNDS GENELABS TECHNOLOGIES, INC. (US) 2008-10-08 EP claimed
US-20070265262-A1 N-(6-MEMBERED AROMATIC RING)-AMIDO ANTI-VIRAL COMPOUNDS GENELABS TECHNOLOGIES, INC. 2007-11-15 US claimed
WO-2007070556-A2 N-(6-MEMBERED AROMATIC RING)-AMIDO ANTI-VIRAL COMPOUNDS GENELABS TECHNOLOGIES, INC. (US) 2007-06-21 WO claimed
US-20050130251-A1 Reagent for determination of hydrogen peroxide KYOWA MEDEX CO., LTD. (JP) 2005-06-16 US claimed
EP-1424554-A1 REAGENT FOR DETERMINING HYDROGEN PEROXIDE KYOWA MEDEX CO., LTD. (JP) 2004-06-02 EP claimed
US-9095565-B2 Methods for treating blood disorders PHOENICIA BIOSCIENCES, INC. (US) 2015-08-04 US disclosed
US-20140301975-A1 Methods for Treating Blood Disorders PHOENICIA BIOSCIENCES INC (US) 2014-10-09 US disclosed
US-8759378-B2 Methods for treating blood disorders PHOENICIA BIOSCIENCES, INC. (US) 2014-06-24 US disclosed
CN-103420923-A 4-aminoquinazolinehydroxamic acid compounds and applications thereof as antitumor medicaments SINOPHARM YIXIN PHARMACEUTICAL CO LTD 2013-12-04 CN disclosed
CN-101857588-B 4-aromatic aminoquinazoline derivative and purpose thereof UNIV SOUTHEAST 2013-11-27 CN disclosed
US-20050130251-A1 Reagent for determination of hydrogen peroxide KYOWA MEDEX CO., LTD. (JP) 2005-06-16 US disclosed
WO-2005023807-A2 4 - HETEROBICYCLYAMINO - SUBSTITUTED QUINAZOLINES AND ANALOGUES THEROF AS CAPSAICIN - ANTAGONISTS NEUROGEN CORPORATION (US) 2005-03-17 WO disclosed
EP-1424554-A1 REAGENT FOR DETERMINING HYDROGEN PEROXIDE KYOWA MEDEX CO., LTD. (JP) 2004-06-02 EP disclosed
WO-1994011365-A1 SUBSTITUTED BENZIMIDAZOLES AND QUINAZOLINES AS ANTIHYPERTENSIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1994-05-26 WO disclosed
US-4808715-A HYPERTENSIVE AGENTS JOHN WYETH & BROTHER LIMITED (GB) 1989-02-28 US disclosed
US-4062844-A Process for preparing hypotensive 2-(4-aroylpiperazin-1-yl)-amino-6,7-dimethoxyquinazolines PFIZER INC. (US) 1977-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070265262-A1 N-(6-MEMBERED AROMATIC RING)-AMIDO ANTI-VIRAL COMPOUNDS ZC3HAV1, HAVCR2, ZC3HAV1L PI4KA 4153/4885PI4K2B 3879/4885PI4K2A 4065/4885
US-20140301975-A1 Methods for Treating Blood Disorders HBB, HBG1, HBG2 PI4KA 4767/4885PI4K2B 4657/4885PI4K2A 4597/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.