SCHEMBL2010261

SCHEMBL2010261

CC(C)(C)OC(=O)[C@H]1NSC(=O)C1=O

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
GAA P10253 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010600 1.00 MAPK1 (0.35) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL19520662 0.64 MAPK1 (0.41) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL21854629 0.63 MAPK1 (0.37) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL2155137 0.62 MAPK1 (0.36) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL2011204 0.61 MAPK1 (0.36) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL23007075 0.61 NFKB1 (0.38) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL27760177 0.61 MAPK1 (0.38) MAPK1GAA
SCHEMBL321152 0.60 MAPK1 (0.44) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL17962577 0.60 MAPK1 (0.37) MAPK1NFKB1NFKB2RELAGAA
SCHEMBL14718807 0.59 MAPK1 (0.40) MAPK1NFKB1NFKB2RELAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011067266-A1 CARBOXYLIC ACID ANALOGS AS GLYCOGEN SYNTHASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-09 WO disclosed