SCHEMBL20103030

SCHEMBL20103030

CCc1cc(OC)c2nc(N)sc2c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.54
TDP1 Q9NUW8 1/20 0.54
SMN1; SMN2 Q16637 4/20 0.50
RAB9A P51151 3/20 0.50
NPC1 O15118 2/20 0.50
PTGS2 P35354 1/20 0.44
ALDH1A1 P00352 6/20 0.42
HSD17B10 Q99714 2/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
HPGD P15428 1/20 0.38
NSD1 Q96L73 1/20 0.37
TP53 P04637 2/20 0.37
TSHR P16473 2/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103032 0.88 CYP3A4 (0.54) CYP3A4TDP1SMN1; SMN2RAB9ANPC1
SCHEMBL28071115 0.80 CYP3A4 (0.47) CYP3A4TDP1SMN1; SMN2RAB9ANPC1
SCHEMBL29803040 0.80 CYP3A4 (0.60) CYP3A4TDP1SMN1; SMN2RAB9AALDH1A1
SCHEMBL28795289 0.80 CYP3A4 (0.60) CYP3A4TDP1SMN1; SMN2RAB9AALDH1A1
SCHEMBL9722840 0.79 CYP3A4 (0.58) CYP3A4TDP1SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL2664863 0.79 HSD17B10 (0.64) CYP3A4TDP1SMN1; SMN2RAB9AALDH1A1
SCHEMBL4128702 0.78 NPC1 (0.42) CYP3A4TDP1SMN1; SMN2RAB9ANPC1
SCHEMBL24347816 0.78 ALDH1A1 (0.62) CYP3A4SMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL21054913 0.78 NSD1 (0.58) CYP3A4TDP1SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL21091722 0.78 CYP3A4 (0.57) CYP3A4TDP1SMN1; SMN2RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081276-A1 COMPOUNDS TESARO, INC. (US) 2018-05-03 WO disclosed