SCHEMBL20103532

SCHEMBL20103532

COC(=O)C(C)(F)[C@H](c1cccc(CO)c1)C1CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 5/20 0.46
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
CTRB1 P17538 1/20 0.35
SMYD3 Q9H7B4 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CHRM3 P20309 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
HPGDS O60760 1/20 0.33
EPHX1 P07099 1/20 0.33
PRKCA P17252 1/20 0.32
PRKCD Q05655 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21688303 1.00 FFAR1 (0.46) FFAR1PDK1PDK2PDK3PDK4
SCHEMBL20103560 0.89 FFAR1 (0.44) FFAR1CTRB1MEN1KMT2AEPHX1
SCHEMBL21644939 0.88 FFAR1 (0.49) FFAR1PDK1PDK2PDK3PDK4
SCHEMBL21644942 0.88 FFAR1 (0.49) FFAR1PDK1PDK2PDK3PDK4
SCHEMBL20103648 0.85 FFAR1 (0.41) FFAR1CTRB1MEN1KMT2A
SCHEMBL20103443 0.84 FFAR1 (0.44) FFAR1
SCHEMBL20103446 0.84 FFAR1 (0.44) FFAR1
SCHEMBL20103527 0.84 FFAR1 (0.44) FFAR1
SCHEMBL20103672 0.83 FFAR1 (0.57) FFAR1PDK1PDK2PDK3PDK4
SCHEMBL21688395 0.83 FFAR1 (0.43) FFAR1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081047-A1 CYCLOHEXYL GPR40 AGONISTS FOR THE TREATMENT OF TYPE II DIABETES JANSSEN PHARMACEUTICA NV (BE) 2018-05-03 WO disclosed