SCHEMBL20105164

SCHEMBL20105164

Cc1nc(N)cn(C)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.37
TTK P33981 1/20 0.37
AURKB Q96GD4 1/20 0.37
INCENP Q9NQS7 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
BRD4 O60885 9/20 0.36
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
HPGD P15428 3/20 0.36
GLA P06280 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20614414 0.77 ALDH1A1 (0.38) AURKATTKAURKBINCENPBRD4
SCHEMBL13074741 0.74 BRD4 (0.41) BRD4ALDH1A1KDM4EHPGDGLA
SCHEMBL19869652 0.74 BRD4 (0.42) AURKATTKAURKBINCENPBRD4
SCHEMBL5366019 0.72
SCHEMBL20105210 0.71 BRD4 (0.35) BRD4ALDH1A1KDM4EHPGDGLA
SCHEMBL12157416 0.71 BRD4 (0.35) BRD4ALDH1A1KDM4EHPGDGLA
SCHEMBL18073640 0.71 BRD4 (0.35) NOS3NOS1NOS2BRD4ALDH1A1
Hydrochloric Acid SCHEMBL14912306 0.70
SCHEMBL25659106 0.70 ADORA2A (0.38) AURKATTKAURKBINCENPBRD4
SCHEMBL16489426 0.69 BRD4 (0.44) BRD4ALDH1A1KDM4EHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3140304-B1 BENZIMIDAZOLE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2018-05-02 EP disclosed