SCHEMBL20105230

SCHEMBL20105230

CN1Cc2cc(F)ccc2C1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 1/20 0.40
OPRM1 P35372 2/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 2/20 0.39
DPP4 P27487 4/20 0.37
DPP8 Q6V1X1 3/20 0.37
DPP9 Q86TI2 3/20 0.37
PITRM1 Q5JRX3 1/20 0.37
PGR P06401 2/20 0.36
KCNH2 Q12809 2/20 0.36
TMEM97 Q5BJF2 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
DPP7 Q9UHL4 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HSP90B1 P14625 2/20 0.35
TRAP1 Q12931 2/20 0.35
KDM1A O60341 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1950822 0.78 MAPT (0.35) ALDH1A1
SCHEMBL31082076 0.78 BRD4 (0.44) SRD5A1DPP8DPP9PGRDPP7
SCHEMBL14649682 0.75 ALDH1A1 (0.37) SIGMAR1ALDH1A1
SCHEMBL30232454 0.74 DPP4 (0.46) SRD5A1OPRM1OPRK1OPRL1DPP4
SCHEMBL1952644 0.73 TDP2 (0.44) DPP7ALDH1A1L3MBTL1
SCHEMBL18559550 0.72 HTR2A (0.39) OPRM1
SCHEMBL31394041 0.70 ROCK1 (0.39)
SCHEMBL8228638 0.70 DPP9 (0.47) DPP4DPP8DPP9PITRM1KCNH2
SCHEMBL20618318 0.69 SLC6A2 (0.35) PGRSLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL1950736 0.68 KDM4E (0.35) OPRM1OPRK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3140304-B1 BENZIMIDAZOLE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2018-05-02 EP disclosed