SCHEMBL20108094

SCHEMBL20108094

O=C(O)c1ccc(Br)c(F)c1OCC(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 5/20 0.36
TAS2R14 Q9NYV8 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
HSD17B10 Q99714 3/20 0.35
TSHR P16473 2/20 0.35
HPGD P15428 2/20 0.35
NPSR1 Q6W5P4 3/20 0.35
MEN1 O00255 2/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
S1PR2 O95136 1/20 0.35
S1PR4 O95977 1/20 0.35
GAA P10253 1/20 0.35
XBP1 P17861 1/20 0.35
PAX8 Q06710 1/20 0.35
S1PR3 Q99500 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20107976 0.88 KDM4E (0.38) L3MBTL1KDM4EALDH1A1SMN1; SMN2TSHR
SCHEMBL5604030 0.84 L3MBTL1 (0.41) L3MBTL1KDM4EALDH1A1TAS2R14SMN1; SMN2
SCHEMBL31535215 0.77 THRA (0.50) L3MBTL1KDM4EALDH1A1MEN1KMT2A
SCHEMBL30316357 0.77 HSD17B10 (0.50) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL7559576 0.76 SMN1; SMN2 (0.40) L3MBTL1KDM4EALDH1A1TAS2R14SMN1; SMN2
SCHEMBL29816669 0.75 DHODH (0.38) KDM4EALDH1A1TAS2R14HSD17B10TSHR
SCHEMBL20108093 0.75 DHODH (0.38) KDM4EALDH1A1TAS2R14HSD17B10TSHR
SCHEMBL21853468 0.75 DHODH (0.38) KDM4EALDH1A1TAS2R14HSD17B10TSHR
SCHEMBL7554664 0.74 SCN9A (0.35) L3MBTL1KDM4EALDH1A1TAS2R14MEN1
SCHEMBL6600427 0.73 FABP3 (0.47) L3MBTL1KDM4EALDH1A1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3532468-B1 2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH BAYER AG (DE) 2022-03-23 EP disclosed
WO-2018077923-A1 2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH BAYER AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed