SCHEMBL20108430

SCHEMBL20108430

Cc1cc(F)c(-c2ccc(CC(C)(C)C)cc2)c(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
KIF11 P52732 7/20 0.38
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
AR P10275 1/20 0.31
NR3C1 P04150 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26373608 0.78 AR (0.41) ESR1CYP11B1CYP11B2ARAKR1C3
SCHEMBL18272234 0.75 HTR2A (0.39) KIF11CYP11B1CYP11B2AR
SCHEMBL20108617 0.74 CYP11B1 (0.38) KIF11CYP11B1CYP11B2ARAKR1C3
SCHEMBL26373461 0.73 ESR1 (0.41) ESR1KIF11ARRXRARXRB
SCHEMBL24513805 0.73 CYP11B1 (0.39) KIF11CYP11B1CYP11B2AR
SCHEMBL20108522 0.72 APP (0.34) KIF11CYP11B1CYP11B2AKR1C3AKR1C2
SCHEMBL25844613 0.71 AR (0.49) CYP11B1CYP11B2ARAKR1C3AKR1C2
SCHEMBL12142093 0.71 KIF11 (0.50) ESR1KIF11CYP11B1CYP11B2
SCHEMBL2600031 0.71 PTPN7 (0.47) ESR1KIF11AR
SCHEMBL20108386 0.67 AR (0.45) CYP11B1CYP11B2ARAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964635-B1 ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2018-05-02 EP disclosed