SCHEMBL20108451

SCHEMBL20108451

Brc1ccc(SN2CCOCC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
MGLL Q99685 2/20 0.47
CYP1A1 P04798 1/20 0.44
CYP1B1 Q16678 1/20 0.44
POLB P06746 1/20 0.41
AKR1C3 P42330 1/20 0.41
PHGDH O43175 1/20 0.40
HSD17B10 Q99714 3/20 0.40
MAPT P10636 4/20 0.39
PKM P14618 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
ALDH1A1 P00352 3/20 0.38
LMNA P02545 3/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 2/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MPI P34949 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11798954 0.89 MGLL (0.48) KMT2AMEN1MGLLPOLBHSD17B10
SCHEMBL20311368 0.81 MAOB (0.38) KMT2AMEN1MGLLPOLBNPC1
SCHEMBL19903214 0.81 HPGD (0.39) KMT2AMEN1NPC1RAB9AALDH1A1
SCHEMBL24894095 0.80 SMN1; SMN2 (0.49) KMT2AMEN1MGLLPOLBAKR1C3
SCHEMBL24893972 0.80 FKBP1A (0.49) MGLLAKR1C3PHGDHHSD17B10MAPT
SCHEMBL17974492 0.80 MGLL (0.39) KMT2AMEN1MGLLPOLBHSD17B10
SCHEMBL24893956 0.80 MAPT (0.41) KMT2AMGLLAKR1C3PHGDHHSD17B10
SCHEMBL19903237 0.79 HPGD (0.38) KMT2AMEN1MGLLHSD17B10MAPT
SCHEMBL9579555 0.79 MAPT (0.49) KMT2AMEN1MGLLPOLBHSD17B10
SCHEMBL19478738 0.78 SMN1; SMN2 (0.47) KMT2AMEN1MGLLPOLBAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed
EP-2976339-B1 GEMINALLY SUBSTITUTED CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-06-27 EP disclosed
EP-2976340-B1 CYCLOALKYL NITRILE PYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-06-13 EP disclosed
EP-2964635-B1 ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2018-05-02 EP disclosed