SCHEMBL20110031

SCHEMBL20110031

C=CCCc1nccc(CC)n1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
CYP1A2 P05177 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16248159 0.80 KDM4E (0.37) CYP1A2POLB
SCHEMBL830187 0.77 CYP1A2 (0.37) CYP1A2POLB
Ammonia Solution, Strong SCHEMBL28652832 0.75 CYP1A2 (0.36) CYP1A2POLB
Ammonia Solution, Strong SCHEMBL11451734 0.74 CYP1A2 (0.35) CYP1A2POLB
SCHEMBL28806573 0.72 MAP4K4 (0.35) CYP1A2POLB
SCHEMBL28160853 0.72 CYP1A2 (0.38) CYP1A2POLB
SCHEMBL25987002 0.72 SORD (0.47) CYP1A2POLB
Formamide SCHEMBL29265659 0.71 CYP1A2 (0.35) CYP1A2POLB
SCHEMBL12313633 0.71 NOS3 (0.30)
SCHEMBL16015473 0.71 HRH3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed