SCHEMBL20116291

SCHEMBL20116291

Cc1ccc2cnc(Br)n2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
KDM4E B2RXH2 5/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 4/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
APP P05067 1/20 0.32
PAX8 Q06710 1/20 0.32
CHEK1 O14757 1/20 0.32
LIMK1 P53667 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15833696 0.79 CYP1A2 (0.40) CYP1A2CYP2C9KDM4ENPC1RAB9A
SCHEMBL21611244 0.72 CYP1A2 (0.35) CYP1A2CYP2C9KDM4ENPC1RAB9A
SCHEMBL16158619 0.69 KDM4E (0.37) CYP1A2CYP2C9KDM4ENPC1RAB9A
SCHEMBL31479337 0.68 KDM4E (0.35) KDM4ENPC1RAB9AMAPK1ALDH1A1
SCHEMBL13676388 0.68 CYP1A2 (0.53) CYP1A2CYP2C9KDM4ENPC1RAB9A
SCHEMBL10207538 0.67 KDM4E (0.58) KDM4ENPC1RAB9AMAPK1ALDH1A1
SCHEMBL32664927 0.63 RAB9A (0.48) KDM4ENPC1RAB9AMAPK1ALDH1A1
SCHEMBL10238918 0.63 CYP1A2 (0.56) CYP1A2CYP2C9KDM4ENPC1RAB9A
SCHEMBL19631265 0.63 KDM4E (0.33) CYP1A2KDM4ENPC1RAB9AMAPK1
SCHEMBL22300408 0.62 CYP1A2 (0.50) CYP1A2CYP2C9KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed