SCHEMBL20116484

SCHEMBL20116484

CCOc1cnc(C#N)cc1NC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.44
SRC P12931 3/20 0.38
LMNA P02545 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
GRM5 P41594 1/20 0.36
CTSS P25774 1/20 0.36
STK4 Q13043 3/20 0.35
STK3 Q13188 1/20 0.35
HSD17B10 Q99714 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
EGFR P00533 2/20 0.35
ERBB2 P04626 2/20 0.35
PDE4D Q08499 1/20 0.34
GAA P10253 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20676395 0.79 CHEK1 (0.40) CHEK1LMNACYP1A2CYP3A4GRM5
SCHEMBL20117027 0.78 PDE4A (0.42) CHEK1SRCLMNACTSSKDM4E
SCHEMBL21749932 0.78 PDE4A (0.43) CHEK1SRCLMNAKDM4EALDH1A1
SCHEMBL21045855 0.75 CHEK1 (0.40) CHEK1LMNACYP1A2CYP3A4GRM5
SCHEMBL30439920 0.75 CHEK1 (0.40) CHEK1LMNACYP1A2CYP3A4GRM5
SCHEMBL29040356 0.74 KDM4E (0.38) CHEK1CYP1A2GRM5CTSSHSD17B10
SCHEMBL20929469 0.72 JAK2 (0.40) CHEK1SRC
SCHEMBL21045740 0.71 LTA4H (0.47) CHEK1CTSSGAASLC6A2SLC6A4
SCHEMBL30439893 0.71 LTA4H (0.47) CHEK1CTSSGAASLC6A2SLC6A4
SCHEMBL21045796 0.70 AR (0.44) CHEK1CYP1A2CYP3A4CTSSKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed