SCHEMBL29040356

SCHEMBL29040356

CCOc1cnc(C#N)cc1COC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 5/20 0.38
HPGD P15428 5/20 0.38
HSD17B10 Q99714 4/20 0.38
CHEK1 O14757 3/20 0.38
GAA P10253 1/20 0.37
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
MAPK1 P28482 1/20 0.35
CTSS P25774 1/20 0.34
CYP1A2 P05177 1/20 0.34
TRPV4 Q9HBA0 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117027 0.79 PDE4A (0.42) KDM4EALDH1A1HPGDCHEK1GAA
SCHEMBL21749932 0.79 PDE4A (0.43) KDM4EALDH1A1HPGDCHEK1GAA
SCHEMBL20676395 0.77 CHEK1 (0.40) KDM4EALDH1A1HPGDHSD17B10CHEK1
SCHEMBL21097993 0.76 KDM4E (0.38) KDM4EALDH1A1HPGDHSD17B10CHEK1
SCHEMBL20116484 0.74 CHEK1 (0.44) KDM4EALDH1A1HSD17B10CHEK1GAA
SCHEMBL21045855 0.72 CHEK1 (0.40) KDM4EALDH1A1HSD17B10CHEK1PDE4A
SCHEMBL30439920 0.72 CHEK1 (0.40) KDM4EALDH1A1HSD17B10CHEK1PDE4A
SCHEMBL21045740 0.69 LTA4H (0.47) HPGDCHEK1GAACTSSCSF1R
SCHEMBL30439893 0.69 LTA4H (0.47) HPGDCHEK1GAACTSSCSF1R
SCHEMBL21045796 0.68 AR (0.44) KDM4ECHEK1CTSSCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117777121-A Compounds and uses thereof 詹森药业有限公司 2024-03-29 CN disclosed
CN-110099898-B Compounds and uses thereof 优曼尼蒂治疗公司 2023-07-25 CN disclosed