SCHEMBL20116490

SCHEMBL20116490

CCOC(=N)c1ccc(OC)c(N)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.57
PDE4B Q07343 3/20 0.57
PDE4C Q08493 3/20 0.57
PDE4D Q08499 3/20 0.57
ALDH1A1 P00352 3/20 0.57
LMNA P02545 1/20 0.57
HTT P42858 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
CYP3A4 P08684 1/20 0.50
TUBB4A P04350 1/20 0.49
TUBB P07437 1/20 0.49
TUBA3C P0DPH7 1/20 0.49
TUBA1B P68363 1/20 0.49
TUBA4A P68366 1/20 0.49
TUBB4B P68371 1/20 0.49
TUBB3 Q13509 1/20 0.49
TUBB2A Q13885 1/20 0.49
TUBB8 Q3ZCM7 1/20 0.49
TUBA3E Q6PEY2 1/20 0.49
TUBA1A Q71U36 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116214 0.84 PRSS1 (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL12287386 0.82 DGAT1 (0.50) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL1300394 0.82 HSD17B2 (0.65) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL20116491 0.81 PDE4B (0.56) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL9219136 0.77 DGAT1 (0.53) ALDH1A1LMNAL3MBTL1USP2PRSS1
SCHEMBL21823575 0.76 PRSS1 (0.54) PDE4APDE4BPDE4CPDE4DHSD17B10
Hydrochloric Acid SCHEMBL2461112 0.75 HSD17B2 (0.45) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL27014428 0.75 PRKCI (0.54) ALDH1A1HTTGAAPRSS1DGAT1
SCHEMBL13108706 0.75 DGAT1 (0.62) ALDH1A1LMNAHTTCYP3A4SMN1; SMN2
SCHEMBL11177279 0.75 TSHR (0.63) ALDH1A1CYP3A4NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed