SCHEMBL20116579

SCHEMBL20116579

CCC(C)n1cc2ccc(C)cc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.38
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
NOTUM Q6P988 1/20 0.36
ALDH1A1 P00352 4/20 0.35
ATM Q13315 1/20 0.34
NQO2 P16083 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPT P10636 4/20 0.34
ACHE P22303 2/20 0.34
NLRP3 Q96P20 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
NFKB1 P19838 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SENP8 Q96LD8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117305 0.83 NOTUM (0.43) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL22358039 0.83 PDE10A (0.34) KMT2AMEN1NOTUMALDH1A1MAPT
SCHEMBL20116576 0.78 CYP1A2 (0.41) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL13607533 0.73 NOTUM (0.44) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL422734 0.70 MAPT (0.63) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL12730005 0.69 CYP1A2 (0.41) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL25097119 0.68 CYP1A2 (0.45) CYP1A2KMT2AMEN1ALDH1A1NQO2
SCHEMBL28457711 0.67 HDAC8 (0.37) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL19763359 0.66 NPC1 (0.66) CYP1A2KMT2AMEN1NOTUMALDH1A1
SCHEMBL13607690 0.66 KDM4E (0.42) CYP1A2KMT2AMEN1ALDH1A1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed