SCHEMBL20116576

SCHEMBL20116576

Cc1ccc2cn(C(F)F)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.41
ALDH1A1 P00352 4/20 0.38
NQO2 P16083 1/20 0.37
HDAC4 P56524 2/20 0.37
CYP2A6 P11509 2/20 0.37
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 2/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
NFKB1 P19838 1/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117305 0.84 NOTUM (0.43) CYP1A2ALDH1A1NQO2CYP2A6KMT2A
SCHEMBL20025158 0.79 NPC1 (0.35) ALDH1A1HDAC4KMT2AMAPTMEN1
SCHEMBL16132751 0.79 BACE1 (0.39) CYP1A2ALDH1A1HDAC4CYP2A6KMT2A
SCHEMBL15910725 0.79 KDM4E (0.56) ALDH1A1HDAC4KMT2AMAPTMEN1
SCHEMBL20116579 0.78 CYP1A2 (0.38) CYP1A2ALDH1A1NQO2CYP2A6KMT2A
SCHEMBL29602706 0.73 HDAC8 (0.44) ALDH1A1NQO2HDAC4MAPTKDM4E
SCHEMBL422734 0.73 MAPT (0.63) CYP1A2ALDH1A1NQO2CYP2A6KMT2A
SCHEMBL30147529 0.72 PLK1 (0.43) HDAC4SMN1; SMN2SYK
SCHEMBL25097119 0.72 CYP1A2 (0.45) CYP1A2ALDH1A1NQO2CYP2A6KMT2A
SCHEMBL24873712 0.71 LPL (0.40) HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed