SCHEMBL20116749

SCHEMBL20116749

CC(C)n1ncc2ccc(-c3noc(C4CCN(C=O)CC4)n3)cc21

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.45
HTR4 Q13639 3/20 0.45
SMN1; SMN2 Q16637 6/20 0.42
LMNA P02545 4/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GRM5 P41594 1/20 0.41
KCNH2 Q12809 1/20 0.41
SMO Q99835 1/20 0.41
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PTGER3 P43115 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116813 0.92 NR1H4 (0.43) NR1H4HTR4SMN1; SMN2LMNATSHR
SCHEMBL20676461 0.90 NR1H4 (0.42) NR1H4HTR4SMN1; SMN2LMNATSHR
SCHEMBL20116507 0.86 NR1H4 (0.45) NR1H4HTR4SMN1; SMN2LMNATSHR
SCHEMBL20116846 0.86 NR1H4 (0.45) NR1H4HTR4SMN1; SMN2LMNATSHR
SCHEMBL20117198 0.86 NPC1 (0.54) NR1H4HTR4SMN1; SMN2LMNANPC1
SCHEMBL20116695 0.85 GRM5 (0.35) NR1H4HTR4GRM5PTGER3
SCHEMBL22357882 0.84 SMN1; SMN2 (0.54) NR1H4SMN1; SMN2LMNATSHRHTT
SCHEMBL22357937 0.84 LMNA (0.47) NR1H4SMN1; SMN2LMNATSHRSMO
SCHEMBL22357930 0.84 NR1H4 (0.58) NR1H4HTR4NPC1RAB9AGRM5
SCHEMBL20116409 0.84 GRM5 (0.43) NR1H4HTR4SMN1; SMN2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed