SCHEMBL20117993

SCHEMBL20117993

Nc1cccc2[nH]c3c(c12)CCCCC3

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
EGFR P00533 9/20 0.41
ABL1 P00519 1/20 0.39
ABL2 P42684 1/20 0.39
F2 P00734 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PARP1 P09874 2/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28559488 0.81 SMN1; SMN2 (0.50) SMN1; SMN2KDM4EALDH1A1EGFRPARP1
SCHEMBL28549389 0.81 SMN1; SMN2 (0.50) SMN1; SMN2KDM4EALDH1A1EGFRPARP1
SCHEMBL31447943 0.79 SMN1; SMN2 (0.49) SMN1; SMN2KDM4EALDH1A1EGFRABL1
SCHEMBL11843637 0.77 KDM4E (0.47) SMN1; SMN2KDM4EALDH1A1EGFRF2
SCHEMBL11163975 0.77 ALDH1A1 (0.47) SMN1; SMN2KDM4EALDH1A1EGFRALOX15
SCHEMBL25423026 0.77 NISCH (0.57) KDM4EALOX15HSD17B10PARP1
SCHEMBL28874663 0.74 MAPT (0.47) SMN1; SMN2KDM4EALDH1A1EGFRABL1
SCHEMBL4101907 0.73 HTR2C (0.54) SMN1; SMN2KDM4EALDH1A1EGFRMAPK1
SCHEMBL10736375 0.73 MAPT (0.59) SMN1; SMN2KDM4EALDH1A1PARP1TNKS2
SCHEMBL2485381 0.72 GFER (0.60) SMN1; SMN2KDM4EALDH1A1EGFRALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3315500-A1 FUSED TETRA OR PENTA-CYCLIC DIHYDRODIAZEPINOCARBAZOLONES AS PARP INHIBITORS BeiGene, Ltd. (KY) 2018-05-02 EP disclosed