SCHEMBL2011853

SCHEMBL2011853

CCn1nc(C)cc1C(=O)NCCC(Cc1ccccc1)N(C)C(=O)c1cnc2occc2c1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.59
HCRTR2 O43614 2/20 0.59
STING1 Q86WV6 13/20 0.35
SMYD3 Q9H7B4 2/20 0.35
IRF3 Q14653 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012511 0.87 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL6917571 0.87 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2013624 0.86 HCRTR1 (0.60) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2011420 0.82 HCRTR1 (0.65) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2012845 0.81 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2053609 0.81 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2014719 0.81 HCRTR1 (0.60) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2014489 0.81 HCRTR1 (0.61) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2054242 0.81 HCRTR1 (0.61) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2014566 0.80 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed