SCHEMBL2014719

SCHEMBL2014719

CCn1nc(C)cc1C(=O)NCCC(Cc1ccccc1)N(C)C(=O)c1ccc2ocnc2c1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.60
HCRTR2 O43614 2/20 0.60
STING1 Q86WV6 14/20 0.39
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
GLA P06280 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
IRF3 Q14653 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010859 0.86 HCRTR1 (0.66) HCRTR1HCRTR2CTNNB1WNT3A
SCHEMBL2011853 0.81 HCRTR1 (0.59) HCRTR1HCRTR2STING1ALDH1A1SMYD3
SCHEMBL2011420 0.81 HCRTR1 (0.65) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2013146 0.81 HCRTR1 (0.66) HCRTR1HCRTR2SMYD3
SCHEMBL2051392 0.81 HCRTR1 (0.66) HCRTR1HCRTR2SMYD3
SCHEMBL2053609 0.80 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2012845 0.80 HCRTR1 (0.64) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2013624 0.80 HCRTR1 (0.60) HCRTR1HCRTR2STING1SMYD3IRF3
SCHEMBL2054242 0.80 HCRTR1 (0.61) HCRTR1HCRTR2STING1ALDH1A1CYP1A2
SCHEMBL2014489 0.80 HCRTR1 (0.61) HCRTR1HCRTR2STING1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed