SCHEMBL20121554

SCHEMBL20121554

O=C(CCc1ccc(F)cc1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(Cl)cc2)C1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.68
CYP3A4 P08684 1/20 0.46
MLNR O43193 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
P2RX7 Q99572 1/20 0.40
ME2 P23368 2/20 0.39
ME1 P48163 2/20 0.39
ME3 Q16798 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15760176 0.96 KCNH2 (0.72) KCNH2CYP3A4MLNRP2RX7
SCHEMBL20121572 0.96 KCNH2 (0.72) KCNH2CYP3A4MLNRP2RX7
SCHEMBL20121610 0.95 KCNH2 (0.70) KCNH2CYP3A4MLNRME2ME1
SCHEMBL20121560 0.94 KCNH2 (0.63) KCNH2CYP3A4MLNRP2RX7
SCHEMBL20121576 0.91 KCNH2 (0.78) KCNH2CYP3A4MLNRME2ME1
SCHEMBL20121613 0.91 KCNH2 (0.78) KCNH2CYP3A4MLNRME2ME1
SCHEMBL17636399 0.91 KCNH2 (0.78) KCNH2CYP3A4MLNRME2ME1
SCHEMBL12952054 0.91 KCNH2 (0.70) KCNH2CYP3A4PTGDR2P2RX7
SCHEMBL12951885 0.91 KCNH2 (0.67) KCNH2CYP3A4
SCHEMBL20121570 0.90 KCNH2 (0.64) KCNH2CYP3A4MLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed