SCHEMBL20121603

SCHEMBL20121603

Cc1ccc(Nc2c(-c3ccc(F)cc3)nc3n2CCN(C(=O)CCc2ccc(CN)cc2)C3)cc1

nearest known ligand 0.78

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.78
CYP3A4 P08684 1/20 0.49
MLNR O43193 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
F9 P00740 1/20 0.38
F11 P03951 1/20 0.38
F7 P08709 1/20 0.38
CYP2C9 P11712 1/20 0.38
TGFBR1 P36897 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17636399 0.96 KCNH2 (0.78) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL20121613 0.96 KCNH2 (0.78) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL20121576 0.96 KCNH2 (0.78) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL12952248 0.93 KCNH2 (0.75) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL12952261 0.92 KCNH2 (0.73) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL15760176 0.92 KCNH2 (0.72) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL20121572 0.92 KCNH2 (0.72) KCNH2CYP3A4MLNRMEN1ALDH1A1
SCHEMBL12952250 0.92 KCNH2 (0.75) KCNH2CYP3A4
SCHEMBL20121610 0.91 KCNH2 (0.70) KCNH2CYP3A4MLNR
SCHEMBL12952166 0.91 KCNH2 (0.71) KCNH2CYP3A4MLNRMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed