SCHEMBL20122293

SCHEMBL20122293

CC(C)(C)OC(=O)/N=C(/NCCCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCOc1ccc(CS)c(CS)c1)NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.40
HDAC1 Q13547 3/20 0.40
CA1 P00915 6/20 0.40
CA2 P00918 6/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
SIRT5 Q9NXA8 1/20 0.38
PTPN1 P18031 4/20 0.38
PTPN22 Q9Y2R2 2/20 0.38
CXCR3 P49682 1/20 0.37
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16504795 0.94 HDAC4 (0.42) HDAC4HDAC1CA1CA2ITGB3
SCHEMBL17771363 0.90 CA1 (0.36) HDAC4HDAC1CA1CA2ITGB3
SCHEMBL16521922 0.89 CA1 (0.47) HDAC4HDAC1CA1CA2ITGB3
SCHEMBL16504598 0.84 CA1 (0.45) CA1CA2ITGB3ITGA2BATM
SCHEMBL16504793 0.81 CA12 (0.36) CA1CA2ITGB3ITGA2BCA12
SCHEMBL23626318 0.80 CTSK (0.49) HDAC4HDAC1CA1CA2SIRT5
SCHEMBL16572287 0.78 CTSS (0.48) HDAC4HDAC1CA1CA2SIRT5
SCHEMBL16504607 0.78 CTSS (0.48) HDAC4HDAC1CA1CA2SIRT5
SCHEMBL16572281 0.78 CTSS (0.48) HDAC4HDAC1CA1CA2SIRT5
SCHEMBL16504677 0.78 CTSS (0.48) HDAC4HDAC1CA1CA2SIRT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963427-B2 Dithiol mucolytic agents PARION SCIENCES, INC. (US) 2018-05-08 US disclosed