SCHEMBL20123366

SCHEMBL20123366

COc1cccc(OC)c1/C=C/C(N)=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 4/20 0.67
CYP1A1 P04798 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 1/20 0.56
ALDH1A1 P00352 2/20 0.51
MAPT P10636 2/20 0.51
GAA P10253 1/20 0.51
HTT P42858 1/20 0.51
CYP1B1 Q16678 1/20 0.50
AURKA O14965 1/20 0.49
NFE2L2 Q16236 4/20 0.47
TFEB P19484 1/20 0.47
KDM4E B2RXH2 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BACE1 P56817 2/20 0.46
APP P05067 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3567982 0.85 ABCG2 (0.71) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL3567978 0.85 ABCG2 (0.71) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL16265418 0.83 ABCG2 (0.69) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL16265416 0.83 ABCG2 (0.69) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL16587940 0.83 ABCG2 (0.69) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL6776970 0.81 ABCG2 (0.67) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL3207731 0.81 NFE2L2 (0.67) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL6776974 0.81 ABCG2 (0.67) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL7954649 0.81 ABCG2 (0.67) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1
SCHEMBL3207710 0.81 NFE2L2 (0.67) ABCG2CYP1A1CYP1A2CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2620436-B1 SUBSTITUTED POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVE PRODRUG SHIONOGI & CO (JP) 2018-05-09 EP disclosed