SCHEMBL2012344

SCHEMBL2012344

COC(=O)Oc1c(F)cccc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.44
POLB P06746 1/20 0.44
THRB P10828 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
GLA P06280 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
GPR35 Q9HC97 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27668224 0.85 ALDH1A1 (0.48) HSPB1ALDH1A1MAPTPOLBTSHR
SCHEMBL4090307 0.84 HSPB1 (0.47) HSPB1ALDH1A1MAPTPOLBTHRB
SCHEMBL27796727 0.83 TDP1 (0.51) ALDH1A1MAPTPOLBTSHRKMT2A
SCHEMBL4087050 0.83 HSPB1 (0.46) HSPB1ALDH1A1MAPTPOLBTHRB
SCHEMBL27479661 0.83 HSPB1 (0.48) HSPB1ALDH1A1MAPTPOLBTHRB
SCHEMBL28920607 0.81 HSPB1 (0.47) HSPB1ALDH1A1MAPTTHRBTSHR
SCHEMBL589644 0.80 TDP1 (0.52) HSPB1ALDH1A1MAPTPOLBTSHR
SCHEMBL4087052 0.79 HSPB1 (0.43) HSPB1ALDH1A1MAPTPOLBTSHR
SCHEMBL4087059 0.79 HSPB1 (0.43) HSPB1ALDH1A1MAPTPOLBTSHR
SCHEMBL16388747 0.78 SMN1; SMN2 (0.45) HSPB1ALDH1A1MAPTPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509954-A1 4 -OXO- 1H -QUINOLINE- 3 - CARBOXAMIDES AS MODULATORS OF ATP -BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2012-10-17 EP disclosed
WO-2011072241-A1 4 -OXO- IH -QUINOLINE- 3 - CARBOXAMIDES AS MODULATORS OF ATP -BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-06-16 WO disclosed