SCHEMBL20125007

SCHEMBL20125007

CC(C)c1cc(Cl)c2[nH]c(=O)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.50
CA9 Q16790 4/20 0.50
MAPT P10636 2/20 0.40
THRB P10828 1/20 0.40
F11 P03951 1/20 0.39
EIF4A3 P38919 3/20 0.38
AKR1B1 P15121 2/20 0.35
DAO P14920 1/20 0.35
PDE2A O00408 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33
GSK3B P49841 1/20 0.33
TOP2A P11388 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14828635 0.80 CA12 (0.54) CA12CA9MAPTTHRBF11
SCHEMBL19737508 0.80 CA12 (0.50) CA12CA9MAPTTHRBF11
SCHEMBL19737581 0.79 HDAC4 (0.42) CA12CA9MAPTTHRB
SCHEMBL30022843 0.77 CA12 (0.55) CA12CA9MAPTF11AKR1B1
SCHEMBL12559818 0.77 CA12 (0.55) CA12CA9MAPTF11AKR1B1
SCHEMBL29153243 0.77 CA12 (0.58) CA12CA9MAPTF11AKR1B1
SCHEMBL21729420 0.76 MCL1 (0.44) CA12CA9MAPTTHRBEIF4A3
SCHEMBL19737649 0.76 CA12 (0.36) CA12CA9MAPTTHRBEIF4A3
SCHEMBL31058635 0.75 CA12 (0.56) CA12CA9MAPTF11AKR1B1
SCHEMBL29241812 0.75 CA12 (0.56) CA12CA9MAPTF11AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150675-A1 COMPOUNDS AND USES THEREOF NUVATION BIO INC. (US) 2020-07-23 WO disclosed
EP-3318557-A2 QUINOLONE COMPOUND Otsuka Pharmaceutical Co., Ltd. (JP) 2018-05-09 EP disclosed