SCHEMBL20125014

SCHEMBL20125014

Cc1ccc2nc(-c3ccccn3)nn2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.51
KDM4E B2RXH2 5/20 0.51
GAA P10253 4/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
POLB P06746 2/20 0.51
GLA P06280 1/20 0.51
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
HTT P42858 3/20 0.46
NPSR1 Q6W5P4 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MEN1 O00255 2/20 0.46
AHR P35869 1/20 0.46
TP53 P04637 4/20 0.44
FLT3 P36888 1/20 0.44
PKM P14618 1/20 0.44
MAPK1 P28482 2/20 0.44
NR1H4 Q96RI1 1/20 0.43
GFER P55789 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11468359 0.82 AHR (0.52) MAPTKDM4EGAATDP1AHR
SCHEMBL15828604 0.81 KDM4E (0.42) MAPTKDM4ENPC1RAB9APOLB
SCHEMBL11483589 0.78 HTT (0.47) MAPTKDM4EGAANPC1RAB9A
SCHEMBL10799076 0.78 KDM4E (0.52) MAPTKDM4ENPC1RAB9APOLB
SCHEMBL13750598 0.74 KDM4E (0.46) MAPTKDM4EGAANPC1RAB9A
SCHEMBL14822663 0.72 AHR (0.51) MAPTKDM4EGAAPOLBKMT2A
SCHEMBL7921087 0.69 AHR (0.46) MAPTKDM4EGAANPC1RAB9A
SCHEMBL22889555 0.69 CYP11B2 (0.55) KDM4ENPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL13729698 0.69 KDM4E (0.41) MAPTKDM4EGAANPC1RAB9A
SCHEMBL10987450 0.68 KDM4E (0.52) MAPTKDM4ENPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3318557-A2 QUINOLONE COMPOUND Otsuka Pharmaceutical Co., Ltd. (JP) 2018-05-09 EP disclosed